EGFR
- A8367 AST-1306Summary: EGFR/HER2 inhibitor
- A8366 ARRY-380Target: HER2Summary: Tyrosine kinase HER2 and p95-HER2 inhibitor
- A8365 Varlitinib (ARRY334543)Summary: ErbB inhibitor
- A8357 AG-1478Target: EGFRSummary: EGFR inhibitor,potent and selective
- A8322 Neratinib (HKI-272)3 CitationTarget: EGFRSummary: HER2/EGFR inhibitor,potent and irreversible
- A8319 Dacomitinib (PF299804, PF299)Target: ErbBSummary: HER inhibitor
- A8247 Afatinib (BIBW2992)1 CitationTarget: EGFRSummary: Irreversible EGFR/HER2 inhibitor
- A8234 Erlotinib Hydrochloride2 CitationSummary: Selective EGFR inhibitor
- A8219 Gefitinib (ZD1839)15 CitationTarget: EGFRSummary: Selective EGFR inhibitor
- A8218 Lapatinib7 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible