Bioactive Compounds
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A8441 GSK4613643 CitationTarget: PLKSummary: Plk1 inhibitor -
A8454 Istradefylline (KW-6002)Target: Adenosine A2A ReceptorsSummary: Selective A2A receptor antagonist -
A8456 JTC-801Target: NOP ReceptorsSummary: KOR-3 (NOP) receptor antagonist -
A8504 Pitavastatin Calcium1 CitationTarget: HMG-CoA ReductasesSummary: Enzyme HMGCR inhibitor -
A8518 Rosuvastatin CalciumSummary: HMG-CoA reductase inhibitor -
A8546 R4061 CitationTarget: SykSummary: SYK inhibitor,potent and ATP-competitive -
A8389 Carbenoxolone disodium1 CitationTarget: Gap JunctionsSummary: 11β-HSD inhibitor -
A8422 Emtricitabine1 CitationTarget: Reverse TranscriptasesSummary: Reverse transcriptase inhibitor -
A8553 PTC124 (Ataluren)Summary: CFTR-G542X nonsense allele inhibitor -
A8614 PhortressSummary: Prodrug of antitumor agent 5F 203

