Bioactive Compounds
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B7387 TCS OX2 29Summary: OX2 receptor antagonist -
B7658 TC-SP 14Summary: agonist of Sphingosine-1-Phosphate Receptor 1 (S1P1) -
A4009 CEP-187701 CitationSummary: Proteasome inhibitor -
A4136 TG101348 (SAR302503)2 CitationTarget: FLT3|JAK|c-RETSummary: JAK-2 inhibitor,potent and selective -
A4068 SNX-21121 CitationSummary: Hsp90 inhibitor,ATP-competitve,potent and selective -
A4074 S/GSK1349572Summary: HIV integrase inhibitor, novel and potent -
A4163 UPF 1069Target: PARPSummary: Selective PARP2 inhibitor -
A4031 Telaprevir (VX-950)1 CitationTarget: HCV NS3-4A proteaseSummary: HCV NS3-4A protease inhibitor -
A4095 Pracinostat (SB939)2 CitationTarget: Histone Deacetylases (HDACs)Summary: Pan-HDAC inhibitor -
A4119 AMG-900Summary: Aurora kinase inhibitor
