Bioactive Compounds
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B7594 SalermideSummary: SIRT1 and SIRT2 inhibitor -
B7715 ML 00253764 hydrochlorideSummary: melanocortin MC4 receptor antagonist -
C6524 Laurocapram -
A4137 AZD14802 CitationTarget: JAKSummary: JAK2 inhibitor,ATP-competitive and novel -
A4164 AZD2461Target: PARPSummary: Novel PARP inhibitor -
A4032 VX-222 (VCH-222, Lomibuvir)Target: HCV polymeraseSummary: NNI of HCV RNA polymerase -
A4096 Belinostat (PXD101)3 CitationTarget: Histone Deacetylases (HDACs)Summary: Hydroxamate-type HDAC inhibitor -
A8201 Amprenavir (agenerase)Summary: HIV-1 protease inhibitor -
A4120 MK-5108 (VX-689)1 CitationSummary: Aurora-A kinase inhibitor,highly selective -
A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S proteasome inhibitor
