Bioactive Compounds
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B6684 MK 8861 CitationSummary: A FLAP and PPARα inhibitor, capable of inhibiting leukotriene biosynthesis and inducing apoptosis -
B6730 1400W dihydrochlorideSummary: INOS inhibitor,potent and highly selective -
B6780 DCPIBSummary: volume-sensitive anion channel (VSAC) and and ICl,swell blocker -
B6941 UBP 296Summary: GluR5-subunit containing kainate receptor antagonist -
A2514 Gentamycin Sulfate1 CitationSummary: Aminoglycoside antibiotic -
A8169 Everolimus (RAD001)17 CitationTarget: mTORSummary: MTOR inhibitor -
A2604 CelastrolTarget: ProteasomeSummary: Antioxidant, anti-inflammatory and immunosuppressive agent -
A4089 Mocetinostat (MGCD0103, MG0103)4 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor,isotype-selective and potent -
B5692 Hexa-D-arginine TFASummary: furin inhibitor -
A4413 PD 150606Target: CalpainsSummary: Non-peptide calpain inhibitor

