Bioactive Compounds
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A2548 CarmofurSummary: Cytostatic derivative of fluorouracilm,antineoplatic agent -
A5096 PF-04217903Target: c-METSummary: C-Met inhibitor,selective and ATP-competitive -
A1413 CEP-32496Summary: BRAF(V600E)inhibitor,highly potent -
A8309 Perifosine1 CitationTarget: AktSummary: Akt inhibitor -
A8318 PP242Target: mTORSummary: MTOR inhibitor, selective and ATP-competitive -
A8350 AZD4547Target: FGFRSummary: FGFR inhibitor -
A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: IGF-IR/IR/ALK inhibitor, ATP-competitive -
A8487 Nocodazole8 CitationTarget: Microtubules/TubulinsSummary: microtubule polymerization inhibitor -
A8521 SilodosinSummary: α1-adrenoceptor antagonist -
A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1) inhibitor

