Bioactive Compounds
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B1294 SR-3677Target: ROCKSummary: Rho Kinase (ROCK-II) inhibitor -
B1377 Megestrol AcetateSummary: Anti-estrogen agent -
B1287 Ro 31-8220Target: PKCSummary: pan-PKC inhibitor -
A1078 Large T antigen - rhesus polyomavirus 560-568Summary: Large T antigen -
A4008 MLN22383 CitationSummary: β5 site of the 20S proteasome inhibitor -
A4016 Apoptosis Activator 2Summary: Indoledione caspase activator, cell-permeable -
A4067 RadicicolSummary: ATPase/kinase inhibitor -
A4135 Tofacitinib (CP-690550) Citrate2 CitationTarget: JAKSummary: Potent JAK inhibitor -
A4073 Raltegravir (MK-0518)1 CitationTarget: integraseSummary: HIV-1 integrase inhibitor -
A4161 3-aminobenzamide2 CitationSummary: Potent PARP inhibitor

