Bioactive Compounds
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A4188 2-Methoxyestradiol (2-MeOE2)2 CitationSummary: Apoptotic, antiproliferative and antiangiogenic agent -
A4024 Danoprevir (RG7227)Target: HCV ProteasesSummary: HCV NS3/4A protease inhibitor -
A4094 MC15683 CitationTarget: Histone Deacetylases (HDACs)Summary: Class II HDAC inhibitor,potent and selective -
A4118 Hesperadin1 CitationTarget: Aurora KinasesSummary: Aurora B kinase inhibitor -
A4306 CiprofibrateSummary: PPARα agonist -
A4328 RolipramTarget: Phosphodiesterases (PDEs)Summary: PDE4-inhibitor and an anti-inflammatory agent -
A4395 10-DAB (10-Deacetylbaccatin)Summary: Precursor of antitumor compound Palitaxel and Docetaxel -
A3171 AmadacyclineSummary: Tetracycline antibiotic -
A3320 CO-1686 (AVL-301)1 CitationTarget: EGFRSummary: EGFR inhibitor -
A3330 CP-809101Summary: 5-HT2C receptor agonist

