Bioactive Compounds
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C4894 Thioetheramide-PCSummary: competitive, reversible inhibitor of secretory phospholipase A2 (sPLA2) -
C5316 RWJ 676572 CitationSummary: orally active inhibitor of the MAP kinases p38α and p38β -
B5740 NS 6180Summary: KCa3.1 channel blocker -
B5741 ML 190Summary: κ opioid receptor (KOP) antagonist -
B5765 PF 04885614Summary: NaV1.8 inhibitor -
B6202 L-AP4Summary: group III metabotropic glutamate receptor agonist -
A8893 Rucaparib (free base)1 CitationTarget: PARPSummary: Potent PARP inhibitor -
B8000 GNE-493Summary: Pan-PI3K/mTOR inhibitor -
B8021 GS-7340Summary: HIV reverse transcriptase inhibitor -
B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5 inhibitor

