Bioactive Compounds
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B5904 Regadenoson1 CitationTarget: Adenosine A2A ReceptorsSummary: Highly selective and low affinity A2A adenosine agonist -
B5960 PF-03394197(Oclacitinib)Summary: Novel Janus kinase inhibitor -
B5970 Sanguinarine chlorideSummary: Inhibitor of PP2C and MKP-1 -
A1045 Gap 279 CitationTarget: Gap JunctionsSummary: Selective gap junction blocker -
A4145 TG101209Summary: JAK2/3 inhibitor -
A4529 JW 55Summary: PARP domain inhibitor -
A4453 NSC 687852 (b-AP15)Target: Deubiquitinating enzymes (DUBs)Summary: 19S regulatory particle Inhibitor -
A4484 PRIMA-1METSummary: Restore mutant p53 activity, induce BAX and PUMA -
A3963 A-7696624 CitationSummary: AMPK activator,potent and reversible -
A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2 inhibitor

