Bioactive Compounds
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BA3932 MiriplatinSummary: Miriplatin (SM-11355) is an effective chemotherapeutic agent. -
SL1048 Pregabalin-d4Summary: A stable isotope deuterated compound of Pregabalin -
A8498 PentamidineSummary: Drug to treat protozoal diseases -
A8471 MeticraneSummary: Peripheral-type benzodiazepine receptor (PBR) inhibitor -
B5513 JNJ 5207852 dihydrochlorideSummary: histamine H3 receptor neutral antagonist -
B4856 CAY10603Target: Histone Deacetylases (HDACs)Summary: potent and selective inhibitor of HDAC6 -
B4991 GNE-317Summary: potent, brain-penetrant PI3K inhibitor -
B5953 Dovitinib (TKI258) LactateTarget: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR). -
B5984 Naproxen SodiumSummary: cyclooxygenase inhibitor -
B6054 EAI045Summary: Inhibitor of L858R/T790M EGFR mutants

