Bioactive Compounds
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A8224 StemRegenin 1 (SR1)Summary: AhR antagonist -
A8225 EzatiostatTarget: Gutathione S-transferaseSummary: (GST) P1-1 inhibitor -
A8229 ML161Target: Protease-Activated ReceptorsSummary: PAR1 inhibitor -
A1295 Granisetron HClSummary: 5-HT3 receptor antagonist -
A1450 LidocaineTarget: Histamine H1 ReceptorsSummary: Anasthetic and class Ib antiarrhythmic agent -
A1493 ABT-751 (E7010)1 CitationTarget: Microtubules/TubulinsSummary: Inhibitor of microtubule polymerization,antimitotic -
A1984 Bendamustine HClSummary: Cytostatic agent for non-Hodgkin lymphomas -
A1447 CilnidipineSummary: Blocker of Dual L- and N-type calcium channel -
A1313 GatifloxacinSummary: Fluoroquinolone antibiotic,inhibits bacterial TOPO II -
A1888 TRAM-34Target: Calcium-Activated Potassium (KCa) ChannelsSummary: KCa3.1 blocker,potent and highly selective

