Bioactive Compounds
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B5881 RI-2Target: RAD51Summary: Optimized reversible RAD51 inhibitor -
B5902 LED209Summary: Highly selective for histidine sensor kinase QseC -
B5937 KPT-9274Summary: Orally acitve allosteric inhibitor of PAK4 -
B5983 MN 64Summary: tankyrase inhibitor -
B1282 A 839977Summary: P2X7 antagonist,potent and selective -
B1138 Mps1-IN-2Summary: Mps1 kinase inhibitor -
B1272 FosaprepitantSummary: Neurokinin-1 antagonist -
B2298 Plinabulin (NPI-2358)Target: Vascular Disrupting Agents (VDA)Summary: vascular disrupting agent -
B1969 Mesalamine1 CitationSummary: IKK inhibitor -
B1051 GSK 6503942 CitationTarget: SGKSummary: SGK1 inhibitor

