Bioactive Compounds
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B5892 Nolatrexed (AG-337)Summary: Non-classical thymidylate synthase inhibitor -
B6038 Ozanimod (RPC1063)Summary: agonist of the sphingosine-1-phosphate receptor subtypes 1 and 5 -
B6039 ARQ 621Summary: Eg5 inhibitor -
B1112 Merimepodib1 CitationTarget: IMPDHSummary: Novel noncompetitive inhibitor of IMPDH(Inosine monophosphate dehydrogenase). -
B1382 AnastrozoleTarget: AromatasesSummary: Aromatase inhibitor -
B1212 ImegliminSummary: Antidiabetic agent -
B1007 AVE 09911 CitationTarget: Angiotensin AT1 ReceptorsSummary: Agonist of angiotensin-(1-7) receptor -
B2266 LDE225 (NVP-LDE225,Erismodegib)1 CitationTarget: SmoothenedSummary: Smoothened inhibitor,potent and selective -
B2300 TolvaptanSummary: AVP V2-receptor antagonist -
B1167 Dofequidar fumarateSummary: MDR reversal agent
