Bioactive Compounds
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B2025 Salubrinal1 CitationSummary: Selective eIF2α inhibitor -
B1308 OTSSP167 hydrochlorideSummary: MELK inhibitor,highly potent and selective -
B1162 FRAX5972 CitationTarget: PAKSummary: PAK inhibitor,potent and ATP-competitive -
B1462 KPT-185Summary: CRM1 inhibitor,selective and irrversible -
B1009 Arginase inhibitor 1Summary: Human arginases I and II inhibitor -
B1052 HG-9-91-012 CitationSummary: Pan-SIK (salt-inducible kinases) inhibitor -
B1879 AdipoRonTarget: AdipoR1|AdipoR2Summary: AdipoR1 and AdipoR2 agonist, first orally active -
B1182 ABC294640Target: SKSummary: Sphingosine kinase 2 inhibitor,selective and competitive -
B1286 AZD7545Target: PDHKSummary: PDHK inhibitor,potent and selective -
B1649 RacecadotrilSummary: Potent enkephalinase inhibitor

