Bioactive Compounds
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A3166 AM0953 CitationSummary: Potent LPA1 receptor antagonist -
A3173 MavorixaforTarget: CXCRSummary: CXCR4 antagonist,potent and selective -
A3184 AR-A0144189 CitationTarget: GSK-3Summary: GSK3β inhibitor, ATP-competitive and selective -
A3195 Asunaprevir (BMS-650032)5 CitationSummary: NS3 protease inhibitor -
A3196 AT-101Target: NS3/4a ProteasesSummary: BH3-mimetic,gossypol enantiomer -
A3201 Atrasentan hydrochlorideSummary: Endothelin receptor antagonist -
A3206 AVL-292Summary: Btk inhibitor -
A3210 AZ201 CitationTarget: ATM/ATRSummary: ATR inhibitor,potent and selective -
A3221 Bardoxolone methylTarget: Nrf2Summary: IKK inhibitor, potent antioxidant inflammation modulator -
A3228 BAY 61-3606 dihydrochlorideSummary: Syk tyrosine kinase inhibitor

