Bioactive Compounds
-
A8198 P 22077Summary: USP7/(DUB)USP47 inhibitor -
A2601 Aclacinomycin A4 CitationTarget: TopoisomerasesSummary: Topoisomerase I and II inhibitor -
A4022 BMS-708163 (Avagacestat)Summary: γ-secretase inhibitor -
A4083 Rocilinostat (ACY-1215)5 CitationTarget: Histone Deacetylases (HDACs)Summary: Selective HDAC6 inhibitor -
A4084 Vorinostat (SAHA, MK0683)22 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor -
A4060 Geldanamycin2 CitationSummary: Hsp90 inhibitor,potent and specific -
A4154 Olaparib (AZD2281, Ku-0059436)37 CitationSummary: PARP-1/2 inhibitor -
A4112 Barasertib (AZD1152-HQPA)6 CitationTarget: Aurora KinasesSummary: Aurora Kinase B inhibitor, Potent and selective -
A4036 Sitagliptin phosphate monohydrate10 CitationTarget: DPP-4Summary: Potent DPP-4 inhibitor -
A4230 NSC 66811Summary: MDM2 inhibitor

