Bioactive Compounds
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B7460 GSK 4112Target: Rev-Erb ReceptorsSummary: Rev-Erbα agonist -
B7551 YIL 781Summary: Ghrelin receptor antagonist -
B7735 AS 2034178Summary: GPR40 agonist -
B7743 NKY 80Summary: adenylyl cyclase (AC) inhibitor -
B5020 ICI 174,864Summary: Selective δ opioid antagonist -
A3005 CAL-101 (Idelalisib, GS-1101)8 CitationTarget: PI3KSummary: PI3K inhibitor -
A4013 Aspirin (Acetylsalicylic acid)Summary: Cyclooxygenase (COX) inhibitor -
A4090 JNJ-264815854 CitationTarget: Histone Deacetylases (HDACs)Summary: Potent HDAC inhibitor -
A4062 KW-2478Target: HSP90Summary: Potent Hsp90 inhibitor, novel, non-ansamycin, -
A4077 DabigatranSummary: A potent, reversible direct thrombin inhibitor with core bioactivity of inhibiting thrombus formation.

