Bioactive Compounds
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A8251 TAE684 (NVP-TAE684)Summary: ALK inhibitor,potent and selective -
A2197 DacarbazineTarget: DNA AlkylatingSummary: Antineoplastic( malignant melanoma and sarcomas) -
A2476 Idarubicin HClSummary: Anthracycline and daunorubicin analog,topoisomerase inhibitor -
A2949 Linifanib (ABT-869)Target: VEGFR|PDGFRSummary: VEGFR/PDGFR inhibitor -
A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective -
A2764 PIK-90Summary: PI3K inhibitor,potent selective -
A5354 ZonisamideTarget: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: Antiepileptic with anticonvulsant and mechanistic effect -
A5506 ThiazovivinTarget: ROCKSummary: ROCK inhibitor -
A5391 Varenicline TartrateSummary: Subtype-selective agonist of α4β2 nicotinic receptors,orally active -
A8302 Tenovin-6Target: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT inhibitor and p53 activator
