Bioactive Compounds
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B5778 SA 4503 dihydrochlorideSummary: σ1 receptor agonist -
B5780 UAMC 00039 dihydrochlorideTarget: Dipeptidyl-peptidase IISummary: dipeptidyl peptidase II (DPP-II) inhibitor -
B5039 DCG IVSummary: highly potent agonist for group II mGlu receptors -
B4756 YH239-EESummary: p53-MDM2 antagonist, potent -
B3553 GS-9973Target: SykSummary: Syk inhibitor, orally bioavailable and selective -
B4764 TCS-PIM-1-4aSummary: Pim inhibitor -
B5801 Cyclotraxin BSummary: TrkB receptor antagonist -
B6263 L-CCG-lllSummary: inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate. -
A3005 CAL-101 (Idelalisib, GS-1101)8 CitationTarget: PI3KSummary: PI3K inhibitor -
A4013 Aspirin (Acetylsalicylic acid)Summary: Cyclooxygenase (COX) inhibitor
