Bioactive Compounds
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A3744 QuetiapineTarget: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptorSummary: Dopamine receptor antagonist -
A3752 Reparixin1 CitationTarget: CXCRSummary: Inhibitor of CXCL8 receptor and CXCR1/CXCR2 activation -
A3761 RG2833Target: HDACSummary: Brain-penetrant HDAC inhibitor -
A3762 RG71125 CitationTarget: MDM2Summary: MDM2 inhibitor, first clinical -
A3766 Rimonabant hydrochlorideSummary: CB1 receptor inverse agonist -
A3785 SalinomycinTarget: AntibioticSummary: Polyether ionophore antibiotic;anti-cancer -
A3808 SD-208Summary: TGF-βR I kinase inhibitor -
A3889 Trelagliptin succinateSummary: DPP-4 inhibitor -
A3901 UNC12151 CitationTarget: L3MBTLSummary: Chemical probe for the methyllysine (Kme) -
A3943 XMD8-92Target: ERKSummary: BMK1/ERK5 inhibitor

