Bioactive Compounds
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A5489 Zibotentan (ZD4054)1 CitationSummary: ETA receptor antagonist,potent and specific -
A5566 LY22288201 CitationTarget: p38Summary: P38 MAP kinase inhibitor -
A5854 Dapagliflozin1 CitationSummary: SGLT2 inhibitor,potent and selective -
A5880 R406 (free base)Summary: Syk inhibitor -
A5970 IrbesartanTarget: Angiotensin AT1 ReceptorsSummary: Angiotensin II inhibitor -
A1986 Nu 6027Target: Cyclin-Dependent Kinases|ATM/ATRSummary: ATR/CDK inhibitor, potent and selective -
A2173 SC 1441 CitationTarget: GlycoproteinsSummary: Gp130 inhibitor -
A8330 CX-4945 (Silmitasertib)13 CitationSummary: CK2 inhibitor -
A8336 KU-600192 CitationTarget: ATM/ATRSummary: ATM kinase inhibitor,potent and selective -
A8339 TAK-875Target: GPR40Summary: GPR40 agonist

