Signaling pathways
- BA2853 MSN-125Summary: MSN-125 is a potent and oligomerization inhibitor.
- BA2854 BTT-3033Summary: BTT-3033 is an orally active conformation-selective (130nM) inhibitor that binds to the α2Idomain.
- BA2855 FasentinSummary: Fasentin is a potent glucose uptake inhibitor that inhibits transport proteins.
- BA2856 MI-1061Summary: MI-1061 is a potent, orally bioavailable, chemically stable (MDM2-p53 interactions) inhibitor.
- BA2857 CurzereneSummary: Curzerene is a sesquiterpene, isolated from the rhizome of Gaertn, which has anticancer activity.
- BA2858 MC4033Summary: MC4033 is a selective, reversible inhibitor of lysine acetyltransferase 8.
- BA2859 BJE6-106Summary: BJE6-106 (B106) is a potent and selective inhibitor.
- BA2861 InecalcitolSummary: Inecalcitol (TX522), a unique vitamin D3 analog, is an orally active vitamin D receptor agonist.
- BA2862 ForodesineSummary: Forodesine (BCX-1777) is a potent, orally active purine nucleoside phosphorylase inhibitor with values ranging from 0.48 to 1.57 nM in humans, mice, rats, monkeys and dogs.
- BA2863 WDR5-IN-1Summary: WDR5-IN-1 is a potent and selective WD repeat structural domain 5 inhibitor.