Biochemical Reagent
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BA5498 ML380Summary: ML380 is a potent, subtype-selective and blood-brain-barrier-crossing orthosteric modulator (PAM) with values of 190 and 610 nM for human and rat M5, respectively. -
BA5499 PentoxyverineSummary: An orally active sigma-1 receptor agonist and muscarinic receptor antagonist with potent antitussive activity -
BA5501 SolifenacinSummary: Solifenacin is a novel muscarinic receptor antagonist. -
BA5502 ImidafenacinSummary: Imidafenacin (KRP-197; ONO-8025) is a potent and selective M3 receptor inhibitor. -
BA5503 DarifenacinSummary: A selective M3 muscarinic receptor antagonist for urinary incontinence and cancer mechanisms -
BA5504 PQCASummary: PQCA is a highly selective and potent modulator of muscarinic receptor-positive mutations. -
BA5505 JHU37160Summary: JHU37160 is a potent and permeable agonist across the blood-brain barrier. -
BA5506 AceclidineSummary: An M3 muscarinic acetylcholine receptor modulator and M1 receptor agonist with cycloplegic activity for cholinergic signaling -
BA5507 VU0467485Summary: VU0467485 (AZ13713945) is a potent, selective, orally bioavailable muscarinic acetylcholine receptor 4 orthosteric modulator (PAM). -
BA5508 FustinSummary: Fustinis ((±)-Fustin; 3,7,3',4'-Tetrahydroxyflavanone) is a potent amyloid β inhibitor.

