Protein Tyrosine Kinase/RTK
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C6509 Nilotinib hydrochlorideSummary: An orally active Bcr-Abl tyrosine kinase inhibitor for chronic myeloid leukemia (CML) -
C6401 Chloropyramine hydrochlorideSummary: A histamine H1 receptor antagonist with antiallergic and antitumor applications -
C6375 lenvatinib Mesylate1 CitationSummary: An orally active multi-target tyrosine kinase inhibitor of VEGFR2, VEGFR3, FGFR, and PDGFR for angiogenesis and hepatocellular carcinoma -
C6370 Nintedanib esylateSummary: A triple tyrosine kinase inhibitor of VEGFR, FGFR, and PDGFR -
B8790 TrastuzumabSummary: A humanized monoclonal antibody for the treatment of HER2-positive breast cancer and gastric cancer -
B8781 DeucravacitinibSummary: An orally active TYK2 inhibitor for the treatment of moderate-to-severe plaque psoriasis -
B8391 BLU-554Summary: A highly selective oral FGFR4 inhibitor for the treatment of hepatocellular carcinoma -
B8387 ErdafitinibSummary: An orally available pan-FGFR inhibitor with potential antitumor activity -
B8316 HarmineSummary: Harmine -
B5854 Pexidartinib (PLX3397)7 CitationTarget: FLT3|c-Kit|CSF1RSummary: A multi-targeted receptor tyrosine kinase inhibitor; A CSF-1R inhibitor

