Proteases
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A4426 K 579Summary: Dipeptidyl peptidase IV inhibitor -
A4402 FlurizanSummary: NSAID,inhibits γ-secretase activity -
A4436 GI 254023X2 CitationTarget: ADAMsSummary: Selective inhibitor of ADAM10 metalloprotease -
A8239 CA-074 Me7 CitationTarget: CathepsinsSummary: Cathepsin B inhibitor -
A5066 Heparin sodiumSummary: Antithrombin III activator -
B5856 GSK1349572 sodiuM saltSummary: Next-generation HIV integrase (IN) inhibitor -
C5830 PD 145305Summary: selective inhibitor of calpains -
B7854 o-PhenanthrolineSummary: metalloprotease inhibitor -
A4064 NVP-BEP800Target: HSP90Summary: Oral Hsp90β inhibitor, novel, fully synthetic -
A4031 Telaprevir (VX-950)1 CitationTarget: HCV NS3-4A proteaseSummary: HCV NS3-4A protease inhibitor
