Metabolic Enzyme/Protease
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BA4457 ConvallatoxinSummary: Convallatoxin is a cardiac glycoside isolated from RegeletRadde. -
BA4456 ST247Summary: ST247 is a potent inverse agonist. -
BA4455 BAY-5516Summary: BAY-5516 is an inverse agonist (6.1 ± 3.6 nM). -
BA4453 MavodelparSummary: Mavodelpar (REN001) is a selective agonist. -
BA4451 PTGR2-IN-1Summary: PTGR2-IN-1 is a potent inhibitor. -
BA4450 HWL-088Summary: HWL-088 is a potent, orally active free fatty acid receptor 1 agonist (at 18.9 nM) with moderate activity (at 570.9 nM). -
BA4449 GSK1820795ASummary: GSK1820795A is a selective antagonist as a timosartan analog. -
BA4448 RivoglitazoneSummary: Rivoglitazone is a thiazolidinedione derivative. -
BA4447 GlabroneSummary: Glabrone is an isoflavone isolated from licorice root. -
BA4442 MonascinSummary: Monascin is an azurophilic pigment that can be extracted from red yeast rice and is orally active with antitumor and anti-inflammatory activities.
