Metabolic Enzyme/Protease
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BA4468 F44-A13Summary: F44-A13 is an orally active, highly selective antagonist. -
BA4467 23-epi-26-DeoxyacteinSummary: Natural, orally active compounds with anti-obesity and anti-tumor effects. -
BA4466 NaveglitazarSummary: Naveglitazar (LY519818) is a peroxisome proliferator-activated receptor alpha-gamma dual. -
BA4464 RG-12525Summary: RG-12525 is a specific, competitive, orally available antagonist. -
BA4462 FK614Summary: FK614 is an orally active non-thiazolidinedione (TZD) type selective modulator. -
BA4459 BAY-5094Summary: BAY-5094 is an inverse agonist. -
BA4458 25-Hydroxytachysterol3Summary: 25-Hydroxytachysterol3 is the metabolite. -
BA4457 ConvallatoxinSummary: Convallatoxin is a cardiac glycoside isolated from RegeletRadde. -
BA4456 ST247Summary: ST247 is a potent inverse agonist. -
BA4455 BAY-5516Summary: BAY-5516 is an inverse agonist (6.1 ± 3.6 nM).
