Metabolic Enzyme/Protease
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BA2795 1G244Summary: 1G244 was a potent inhibitor at 12 nM and 84 nM, respectively, but did not inhibit DPPIV and DPPII. - BA2783 BTdCPUSummary: BTdCPU is a heme-regulated inhibitory kinase activator that promotes phosphorylation and induces apoptosis in (Dex)-resistant cancer cells.
- BA2782 JX06Summary: JX06 is a potent, selective, covalent inhibitor.
- BA2778 POMHEXSummary: POMHEX is a racemic mixture of POM precursor active molecules that are cell-permeable and specific inhibitors of HEX.
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BA2763 DinoprostSummary: Dinoprost (ProstaglandinF2α) is an orally effective prostaglandin F (PGF) receptor agonist. - BA2761 KRIBB11Summary: KRIBB11 is an inhibitor.
- BA2755 MilademetanSummary: Milademetan (DS-3032) is a specific, orally active inhibitor for acute myeloid leukemia and solid tumors.
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BA2746 Deferoxamine6 CitationSummary: Deferoxamine (DeferoxamineB) is an iron chelator (binding Fe(III) and many other metal cations) that is widely used to reduce iron accumulation and deposition in tissues. - BA2744 TVB-3166Summary: TVB-3166 is an orally effective, reversible and selective fatty acid synthase inhibitor with 42 nM and 81 nM for FASN and cellular palmitate synthesis, respectively.
- BA2735 HA15Summary: HA15 is a potent and specific inhibitor of endoplasmic reticulum chaperonin.