Signaling Pathways
-
A1736 PA-8241 CitationSummary: Anti-tuberculosis drug -
A2977 Cabozantinib (XL184, BMS-907351)Summary: VEGFR2/Met/Ret/Kit/FLT//AXL inhibitor -
A5092 JNJ-38877605Summary: C-Met inhibitor,ATP-competitive -
A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: Pan-AKT inhibitor,ATP-competitive and potent -
A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective -
A2251 Tivozanib (AV-951)Target: VEGFRSummary: VEGFR inhibitor,potent and selective -
A1266 WYE-354Summary: MTOR inhibitor,potent,ATP-competitive and cell-permeable -
A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ inhibitor -
A2597 Brivanib (BMS-540215)Target: VEGFR|FGFR|Flk1Summary: VEGFR-2 inhibitor,ATP-competitive -
A1630 Epothilone B (EPO906, Patupilone)Target: Microtubules/TubulinsSummary: Microtubule stabilizing macrolide

