Bioactive Compounds
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A4521 TCS PIM-1 1Summary: Pim-1 kinase inhibitor,ATP-competitve -
A4539 NFAT InhibitorSummary: NFAT inhibitor -
A4491 SGC-CBP302 CitationTarget: CREBBP|EP300Summary: Inhibitor of CREBBP/EP300 bromodomain,potent -
A8212 PR-6194 CitationTarget: Deubiquitinating enzymes (DUBs)Summary: Deubiquitylating enzymes (DBUs) inhibitor -
A8216 PP 2 (AG 1879)2 CitationSummary: Src-family kinases inhibitor -
A8251 TAE684 (NVP-TAE684)Summary: ALK inhibitor,potent and selective -
A2197 DacarbazineTarget: DNA AlkylatingSummary: Antineoplastic( malignant melanoma and sarcomas) -
A2476 Idarubicin HClSummary: Anthracycline and daunorubicin analog,topoisomerase inhibitor -
A2949 Linifanib (ABT-869)Target: VEGFR|PDGFRSummary: VEGFR/PDGFR inhibitor -
A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective

