Bioactive Compounds
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A5707 PD318088Target: MEKSummary: Allosteric MEK1/2 inhibitor, non-ATP competitive -
A8386 Busulfan3 CitationSummary: DNA alkylating agent -
A8631 FK 866 HCLTarget: NMPRTaseSummary: NMPRTase inhibitor -
A8691 Flumatinib mesylateSummary: PDGRFβ inhibitor -
A9904 AKT/mTOR Set ISummary: For inhibiting AKT/mTOR -
B1431 (E/Z)-TG003Target: Cdc2-like kinase (Clk)Summary: Cdc2-like kinase (Clk) inhibitor -
B1637 OSI-027Summary: MTORC1/ mTORC2 inhibitor -
B1406 SB5908851 CitationSummary: Potent B-Raf inhibitor -
B1401 Cabozantinib malate (XL184)Summary: MET andVEGF receptor2 inhibitor -
C5813 CFI-400945Summary: orally available, selective inhibitor of polo-like kinase 4 (PLK4)

