Bioactive Compounds
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B8016 UNC20251 CitationTarget: MER|FLT3Summary: orally bioavailable dual MER/FLT3 inhibitor -
B7785 LDN 209929 dihydrochlorideTarget: haspin kinaseSummary: haspin kinase inhibitor -
B4797 HSP990 (NVP-HSP990)Target: HSP90Summary: Hsp90 inhibitor, potent and selective -
B4882 PF-06463922Target: ALK|ROS1Summary: ALK/ROS1 inhibitor,potent and selective -
B4886 DTP3 TFASummary: inhibitor of GADD45β/MKK7 complex -
B4916 GSK 5959Summary: BRPF1 bromodomain inhibitor -
B5822 TMC647055 Choline saltSummary: inhibitor of the hepatitis C virus NS5B polymerase -
B5839 SU66562 CitationTarget: Src|Lyn|YES|FynSummary: Src tyrosine kinases inhibitor -
A1043 Angiotensin III (human, mouse)Summary: Aldosterone stimulator -
B7811 CPI-455 HClSummary: KDM5 inhibitor
