Bioactive Compounds
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A4071 Fluorouracil (Adrucil)12 CitationTarget: Thymidylate SynthaseSummary: Antitumor agent;inhibitor of thymidylate synthase -
A8203 RitonavirSummary: HIV protease inhibitor -
A4121 SNS-314 MesylateTarget: Aurora KinasesSummary: Aurora A/B/C kinases inhibitor, potent and selective -
A4011 ONX-0914 (PR-957)13 CitationTarget: ProteasomeSummary: Immunoproteasome inhibitor,potent and selective -
A4310 Rosiglitazone HClSummary: PPARγ agonist -
A4334 Avanafil1 CitationTarget: Phosphodiesterases (PDEs)Summary: PDE5 inhibitor -
A1915 Zebularine1 CitationTarget: DNA Methyltransferases|Cytidine deaminasesSummary: Cytidine analog; DNA methyltransferase (DNMT) inhibitor; induces DNA demethylation -
A4386 Elesclomol (STA-4783)3 CitationSummary: Oxidative stress/apoptosis inducer,potent and novel -
A3202 Avermectin B1Summary: Insecticide -
A3482 Icotinib HydrochlorideSummary: EGFR inhibitor,potent and specific

