Bioactive Compounds
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B2277 A-803467Target: Voltage-gated Sodium (NaV) ChannelsSummary: NaV1.8 channel blocker,potent and selective -
B1404 DCC-2036 (Rebastinib)Target: FLT3|Bcr-Abl|Tie-2|KDRSummary: Bcr-Abl inhibitor -
B1500 I-BET151 (GSK1210151A)5 CitationTarget: Bromodomain and Extra-Terminal motif (BET)Summary: Selective BET inhibitor -
B1127 UNC 0631Summary: G9a inhibitor -
B5488 BIO-acetoximeSummary: GSK-3α/β inhibitor -
B5508 Alda 12 CitationTarget: Aldehyde DehydrogenasesSummary: ALDH2 activator -
B5516 5'-FluoroindirubinoximeSummary: FMS-like receptor tyrosine kinase-3 (FLT3) inhibitor -
B5527 MM-22Summary: biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide -
B5537 KW 3902Summary: adenosine A1 receptor antagonist -
B5560 Ro 67-7476Summary: positive allosteric modulator of mGlu1 receptors

