Bioactive Compounds
-
A8708 Sephin11 CitationTarget: phosphatasesSummary: Selective PPP1R15A inhibitor -
B5959 GSK J4 free baseSummary: histone demethylase JMJD3/UTX inhibitor -
B5868 MK3102Summary: Novel long-acting DPP-4 inhibitor -
B5954 Dasatinib MonohydrateTarget: PDGFR|c-Kit|Bcr-Abl|SrcSummary: Inhibitor of ABL, SRC, KIT, PDGFR, and other tyrosine kinases. -
C5708 α-Guanidinoglutaric AcidSummary: linear mixed-type inhibitor of nNOS -
C5723 S-(2-aminoethyl) Isothiourea (dihydrobromide)Summary: non-selective inhibitor of all NOS isoforms -
A8764 Rapalink-15 CitationTarget: mTORSummary: third-generation mTOR inhibitor -
L1049 DiscoveryProbe™ Ubiquitination Compound LibrarySummary: A collection of 144 ubiquitination compounds supplied as lyophilized powder or pre-dissolved DMSO solutions -
A1033 [Ser25] Protein Kinase C (19-31)Summary: PKC substrate -
C6532 MES sodium salt

