Bioactive Compounds
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A8883 SAR40533 CitationSummary: Selective ATP-competitive inhibitor of Vps34 -
A8701 Mesoridazine BesylateSummary: Phenothiazine dopamine receptor anatagonist -
B4986 LY2409881Summary: potent and selective IKK2 inhibitor -
B5973 PFI 4Summary: Potent and selective BRPF1 Bromodomain inhibitor -
B6006 NPS-1034Summary: MET inhibitor -
B6026 VR23Target: ProteasomeSummary: proteasome inhibitor -
A5467 Ponatinib (AP24534)1 CitationTarget: VEGFR|PDGFR|Bcr-Abl|FGFR|SrcSummary: pan-BCR-ABL inhibitor,multi-kinase inhibitor -
A5634 SAR245409 (XL765)Summary: mTOR/PI3K inhibitor -
A8321 Cisplatin36 CitationSummary: chemotherapeutic compound -
A8326 AZD-54382 CitationTarget: Cyclin-Dependent KinasesSummary: Potent CDK1/2/9 inhibitor

