Bioactive Compounds
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B5513 JNJ 5207852 dihydrochlorideSummary: histamine H3 receptor neutral antagonist -
B4856 CAY10603Target: Histone Deacetylases (HDACs)Summary: potent and selective inhibitor of HDAC6 -
B4991 GNE-317Summary: potent, brain-penetrant PI3K inhibitor -
B5953 Dovitinib (TKI258) LactateTarget: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR). -
B5984 Naproxen SodiumSummary: cyclooxygenase inhibitor -
B6054 EAI045Summary: Inhibitor of L858R/T790M EGFR mutants -
B1204 Ondansetron hydrochloride dihydrateSummary: 5-HT3 receptor antagonist -
B1709 Clodronate DisodiumSummary: Potent antiosteolytic agent -
B1789 Mexiletine HClTarget: sodium channelSummary: Sodium channel inhibitor -
B1352 BetaxololSummary: βadrenergic receptor blocker

