Bioactive Compounds
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B7335 SB 452533Target: TRPVSummary: TRPV1 antagonist -
A8219 Gefitinib (ZD1839)16 CitationTarget: EGFRSummary: Selective EGFR inhibitor -
A8236 Regorafenib4 CitationTarget: Raf|VEGFR|PDGFR|c-Kit|RETSummary: Inhibitor of VEGFR/PDGFR/FGFR/mutant kit/RET/Raf-1 -
A8246 BEZ235 (NVP-BEZ235)2 CitationSummary: PI3K/mTOR inhibitor,ATP-competitve -
A5118 BTZ043 Racemate2 CitationTarget: DprESummary: DprE1 inhibitor -
A8512 Rifaximin (Xifaxan)Summary: RNA synthesis inhibitor, PXR activator -
A8385 BMS265246Target: Cyclin-Dependent KinasesSummary: CDK1/2 inhibitor,potent and selective -
A8567 Tenovin-3Summary: p53 activator -
A8601 Tankyrase Inhibitors (TNKS) 49Target: TankyrasesSummary: Tankyrase inhibitor -
A9901 Caspase Inhibitor Set ISummary: Caspase Inhibitors

