Bioactive Compounds
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B4754 LDC0000672 CitationTarget: Cyclin-Dependent KinasesSummary: CDK9 inhibitor, novel and highly specific -
B4976 DesogestrelSummary: progestin used in hormonal contraceptives -
B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: inhibitor of VEGFR-2, PDGFRβ, Flt-3, and c-Kit -
B5875 E3330Summary: Ape-1/Ref-1 inhibitor -
B5889 EGF8162 CitationTarget: EGFRSummary: Novel covalent inhibitor of mutant-selective EGFR -
C3503 MS023 (hydrochloride)Summary: type I PRMTs inhibitor -
C4711 AM6545Summary: CB1 selective neutral antagonist -
C4829 UCN-02Summary: protein kinase C inhibitor -
C5557 SR 1824Summary: non-agonist PPARγ ligand -
B1200 PRX-08066Summary: 5-HT2BR antagonist

