Bioactive Compounds
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A1404 Rigosertib sodium salt1 CitationTarget: PLKSummary: Plk1 inhibitor -
A1186 AMG-208Summary: C-Met inhibitor,potent and highly selective -
A2806 BX-912Summary: PDK1 inhibitor,potent and ATP-competitive -
A1718 PosaconazoleTarget: Cytochrome P450 (CYP450)|sterol demethylaseSummary: Sterol C14ɑ demethylase inhibitor -
A2415 AcitretinTarget: RARsSummary: Metabolite of etretinate -
A1987 Ki164256 CitationTarget: LPA ReceptorsSummary: LPA receptor antagonist -
A1352 Zoledronic Acid1 CitationTarget: Farnesyl Diphosphate SynthasesSummary: Potent nitrogen-containing bisphosphonates -
A1778 Vatalanib (PTK787) 2HClTarget: VEGFRSummary: Tyrosine kinase receptor inhibitor -
A5926 FebuxostatSummary: non-purine selective inhibitor of xanthine oxidase -
A5755 MK-17754 CitationSummary: Wee1 kinase inhibtor,potent and ATP-competitive

