Bioactive Compounds
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A1805 Imatinib Mesylate (STI571)2 CitationTarget: PDGFR|c-Kit|Bcr-AblSummary: Abl/c-kit/PDGFR inhibitor -
A1723 Roscovitine (Seliciclib,CYC202)2 CitationSummary: CDK inhibitor,potent and selective -
A2213 17-DMAG (Alvespimycin) HCl1 CitationTarget: HSP90Summary: Hsp90 inhibitor -
A1266 WYE-354Summary: MTOR inhibitor,potent,ATP-competitive and cell-permeable -
A1748 Ramelteon1 CitationTarget: Melatonin ReceptorsSummary: Agonist of melatonin receptor(M1-M2),highly selective -
A2986 ADL5859 HClSummary: δ-opioid receptor agonist,selective -
A1404 Rigosertib sodium salt1 CitationTarget: PLKSummary: Plk1 inhibitor -
A1186 AMG-208Summary: C-Met inhibitor,potent and highly selective -
A2806 BX-912Summary: PDK1 inhibitor,potent and ATP-competitive -
A1718 PosaconazoleTarget: Cytochrome P450 (CYP450)|sterol demethylaseSummary: Sterol C14ɑ demethylase inhibitor

