Bioactive Compounds
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A4194 Obatoclax mesylate (GX15-070)1 CitationTarget: Bcl-2Summary: Potent Bcl-2 inhibitor -
A8202 Abiraterone acetateTarget: Cytochrome P450 (CYP450)Summary: Cytochrome p450 17a1 inhibitor -
A4186 Bromosporine1 CitationTarget: BromodomainsSummary: Bromodomain inhibitor,non-selective -
A4339 AGI-51981 CitationSummary: IDH1 inhibitor against R132 mutant,selective and cell-permeable -
A4364 MethazolamideTarget: Carbonic AnhydrasesSummary: Carbonic anhydrase inhibitor -
A4384 PF-04620110Summary: DGAT-1 inhibitor,potent and selective -
A1921 Z-DQMD-FMK3 CitationTarget: CaspasesSummary: Caspase-3 inhibitor,cell-permeable -
A3198 AT7519 trifluoroacetateSummary: CDK/cyclin inhibitor -
A3199 AT7867 dihydrochlorideSummary: Akt1 and p70S6K/PKA inhibitor -
A3209 AXL1717Target: Insulin-like growth factor receptors(IGFRs)Summary: IGF-1R inhibitor,orally active

