Bioactive Compounds
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B7691 MEDICA 16Summary: Free fatty acid 1 (FFA1/GPR40) receptor agonist -
B7752 GSK 1562590 hydrochlorideSummary: urotensin II (UT) receptor antagonist -
B7765 ML 154Summary: neuropeptide S receptor (NPSR) antagonist -
A2604 CelastrolTarget: ProteasomeSummary: Antioxidant, anti-inflammatory and immunosuppressive agent -
A4089 Mocetinostat (MGCD0103, MG0103)4 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor,isotype-selective and potent -
A4061 IPI-504 (Retaspimycin hydrochloride)3 CitationTarget: HSP90Summary: Hsp90 inhibitor,novel, potent,selective -
A4156 Rucaparib (AG-014699,PF-01367338)3 CitationSummary: Potent PARP inhibitor -
A4168 EntacaponeTarget: Catechol O-Methyltransferase (COMT)Summary: COMT inhibitor -
A4113 ZM 4474392 CitationTarget: Aurora Kinases|MEK|Src|LckSummary: Aurora Kinase inhibitor,potent and selective -
A4037 Vildagliptin (LAF-237)Summary: DPP-4 inhibitor
