Signaling pathways
-
BA8903 DDR2-IN-1Summary: DDR2-IN-1 is a potent inhibitor. - BA8904 GSK-626616Summary: GSK-626616 is a potent orally bioavailable inhibitor.
- BA8905 GNF2133Summary: GNF2133 is a potent, selective, and orally active inhibitor of DYRK1A and GSK3β at 0.0062, >50μM, respectively.
- BA8906 tBIDSummary: tBID is a selective inhibitor of homologous structural domain-interacting protein kinase 2.
- BA8907 DYRK1-IN-1Summary: DYRK1-IN-1 is a highly selective and ligand-efficient inhibitor.
- BA8908 Mirk-IN-1Summary: Mirk-IN-1 (Dyrk1B/A-IN-1) is a highly potent and selective inhibitor of Dyrk1B and Dyrk1A.
- BA8909 AZ-Dyrk1B-33Summary: AZ-Dyrk1B-33 is a potent and selective kinase inhibitor.
- BA8910 Dyrk1A-IN-5Summary: Dyrk1A-IN-5 is a potent and selective inhibitor.
- BA8911 Dyrk1A-IN-4Summary: Dyrk1A-IN-4 is a potent inhibitor with oral activity.
- BA8912 Dyrk1A-IN-3Summary: Dyrk1A-IN-3 is a highly selective bispecific tyrosine-regulated kinase 1A inhibitor that binds DYRK1A with high affinity (=76nM).