Biochemical Reagent
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BA4445 AMG131Summary: AMG131 (INT131) is a potent and highly selective partial agonist that binds to, and replaces, rosiglitazone at ~10nM. -
BA4446 BAY-0069Summary: BAY-0069 is a potent and selective inverse activator at 6.3 nM and 24 nM for human and mouse, respectively. -
BA4452 AdelmidrolSummary: Plays an important anti-inflammatory role. -
BA4454 AleglitazarSummary: Aleglitazar (R1439; RO0728804) is a potent dual agonist with 38nM and 19nM for human and action, respectively. -
BA4460 FTX-6746Summary: FTX-6746 is an orally active inhibitor. -
BA4461 MA-0204Summary: MA-0204 is a potent, highly selective, orally active peroxisome proliferator-activated receptor δ modulator at 0.4 nM, 7.9 nM and 10 nM for human, mouse and rat, respectively. -
BA4463 GSK376501ASummary: GSK376501A is a selective peroxisome proliferator-activated receptor gamma modulator. -
BA4465 EdaglitazoneSummary: Edaglitazone is a potent, selective and orally active agonist. -
BA4469 CRX000227Summary: CRX000227 is a regulator. -
BA4471 CC618Summary: CC618 is a selective peroxisome proliferator-activated receptor antagonist.

