CYP3A/CYP450
- B5724 PentoxyresorufinSummary: fluorometric cytochrome P450 substrate
- B5723 MethoxyresorufinSummary: fluorometric substrate of cytochrome P450
- B5405 YM 511Summary: aromatase (CYP19) inhibitor
- A4322 ClarithromycinTarget: Cytochrome P450 (CYP450)Summary: CYP3A inhibitor, potent
- A4320 VoriconazoleSummary: CYP51 inhibitor
- A4313 Cobicistat (GS-9350)Target: Cytochrome P450 (CYP450)Summary: Selective CYP3A inhibitor
- A3374 DronedaroneTarget: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4 and 2D6 inhibitor,moderate