Bioactive Compounds
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A8618 Palomid 5292 CitationSummary: PI3K/Akt/mTOR inhibitor -
A8629 DBeQTarget: P97 ATPaseSummary: P97 ATPase inhibitor -
B2141 Calcitriol5 CitationSummary: Active metabolite of vitamin D3 -
B2227 BI-D18701 CitationTarget: p90 S6KSummary: P90 RSK inhibitor,ATP-competitive and cell-permeable -
B2277 A-8034672 CitationTarget: Voltage-gated Sodium (NaV) ChannelsSummary: NaV1.8 channel blocker,potent and selective -
B1404 DCC-2036 (Rebastinib)Target: FLT3|Bcr-Abl|Tie-2|KDRSummary: Bcr-Abl inhibitor -
B1500 I-BET151 (GSK1210151A)6 CitationTarget: Bromodomain and Extra-Terminal motif (BET)Summary: Selective BET inhibitor -
C5708 α-Guanidinoglutaric AcidSummary: linear mixed-type inhibitor of nNOS -
C5723 S-(2-aminoethyl) Isothiourea (dihydrobromide)Summary: non-selective inhibitor of all NOS isoforms -
A8764 Rapalink-16 CitationTarget: mTORSummary: third-generation mTOR inhibitor
