Bioactive Compounds
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B7536 PF 998425Summary: non-steroidal androgen receptor (AR) antagonist -
B5174 PKC β pseudosubstrateSummary: Selective cell-permeable peptide inhibitor of protein kinase C -
B5249 PL 017Summary: Selective μ opioid receptor agonist -
B5453 RuBi-4APSummary: voltage-dependent K+ channel blocker -
A5449 PIK-93Summary: PI3Kγ/PI4KIIIβ/PI3Kα inhibitor -
A5455 AEE788 (NVP-AEE788)Summary: EGFR/HER-2/VEGFR inhibitor -
A5511 OfloxacinTarget: Topoisomerases|DNA gyraseSummary: Fluoroquinolones,antibiotics -
A5719 AT7519Target: Cyclin-Dependent KinasesSummary: Multi-CDK inhibitor -
A1947 MEK162 (ARRY-162, ARRY-438162)Target: MEKSummary: MEK1/2 inhibitor,potent and selective -
A8331 Bleomycin Sulfate12 CitationSummary: DNA synthesis inhibitor
