Bioactive Compounds
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A4031 Telaprevir (VX-950)1 CitationTarget: HCV NS3-4A proteaseSummary: HCV NS3-4A protease inhibitor -
A4095 Pracinostat (SB939)2 CitationTarget: Histone Deacetylases (HDACs)Summary: Pan-HDAC inhibitor -
A4119 AMG-900Summary: Aurora kinase inhibitor -
A4234 TW-371 CitationTarget: Bcl-2|Bcl-xl|Mcl-1Summary: Bcl-2 inhibitor, inhibits Bcl-2,Bcl-XL and Mcl-1 -
A4307 GW0742Summary: PPARδ/β agonist,potent and selective -
A4329 CilomilastTarget: Phosphodiesterases (PDEs)Summary: Potent PDE4 inhibitor -
A3177 AN-26901 CitationTarget: AntifungalSummary: Antifungal agent -
A3331 CP-809101 hydrochlorideSummary: 5-HT2C receptor agonist, potent and selective -
A3397 Erlotinib6 CitationSummary: EGFR tyrosine kinase inhibitor -
A3432 GDC-0941 dimethanesulfonateSummary: PI3K inhibitor

