Bioactive Compounds
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A8964 SETDB1-TTD-IN-1Summary: A SETDB1 activator that binds the tandem Tudor domain (TTD) and enhances SETDB1 methyltransferase activity for epigenetic regulation and cancer -
C8544 EGFR/HER2/CDK9-IN-2 -
A9970 cis-Epoxysuccinic acidSummary: An agonist for the succinate receptor (SUCNR1/GPR91) -
SL1032 Rifampicin-d8Summary: A stable isotope deuterated compound of Rifampicin -
BA9141 NRX-103094Summary: NRX-103094 is a potent interaction enhancer with homologous SCF. -
BA3878 CapziminSummary: Capzimin is effective. -
C9053 Rucaparib monocamsylateSummary: A small-molecule PARP inhibitor for research related to DNA repair pathways. -
A4497 PyroxamideTarget: Histone Deacetylases (HDACs)Summary: HDAC1 inhibitor -
A4512 Cucurbitacin I1 CitationTarget: STAT|JAKSummary: STAT3/JAK2 signaling inhibitor -
A5124 Meropenem3 CitationSummary: β-lactam antibiotic of the carbapenem subclass

