Bioactive Compounds
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B7466 NPY 5RA972Summary: neuropeptide Y Y5 receptor antagonist -
B7501 CD 2665Summary: Selective RARβ/γ antagonist -
B7738 SR 35761 CitationTarget: JNKSummary: JNK3 inhibitor, potent and selective -
B6297 Benzoquinonium dibromideSummary: inhibitor of AChR and ganglion -
B6415 CyclothiazideSummary: positive allosteric modulator of AMPA receptors -
B6664 GR 144053 trihydrochlorideSummary: platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonist -
B6716 NF 449Summary: purinergic receptor antagonist -
B6765 Rimcazole dihydrochlorideTarget: Sigma ReceptorsSummary: σ receptors antagonist -
B6814 OLDASummary: endogenous vanilloid TRPV1 (VR1) receptor agonist -
C8598 TPMPA (hydrate)Summary: TPMPA is a selective competitive antagonist for GABAA-ρ (also known as GABAC) receptors, particularly showing selectivity for the ρ1 subtype over ρ2.

